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1

Plant lectins are potent inhibitors of coronaviruses by interfering with two targets in the viral replication cycle

Els Keyaerts, Leen Vijgen, Christophe Pannecouque, Els Van Damme, Willy Peumans, Herman Egberink, Jan Balzarini, Marc Van Ranst

Journal:

Antiviral Research

Year:

2007

Language:

english

File:

PDF, 260 KB

english, 2007

2

Anti-HIV properties of cationic fullerene derivatives

Silvia Marchesan, Tatiana Da Ros, Giampiero Spalluto, Jan Balzarini, Maurizio Prato

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 168 KB

english, 2005

3

Synthesis and anti-HIV Properties of New Water-Soluble Bis-functionalized[60]fullerene Derivatives.

Susanna Bosi, Tatiana Da Ros, Giampiero Spalluto, Jan Balzarini, Maurizio Prato

Journal:

Year:

2004

File:

PDF, 60 KB

2004

4

Aryloxy Phosphoramidate Triesters: a Technology for Delivering Monophosphorylated Nucleosides and Sugars into Cells

Youcef Mehellou, Jan Balzarini, Christopher McGuigan

Journal:

Year:

2009

Language:

english

File:

PDF, 418 KB

english, 2009

5

Structure, physiological role, and specific inhibitors of human thymidine kinase 2 (TK2): Present and future

María-Jesús Pérez-Pérez, Eva-María Priego, Ana-Isabel Hernández, Olga Familiar, María-José Camarasa, Ana Negri, Federico Gago, Jan Balzarini

Journal:

Medicinal Research Reviews

Year:

2008

Language:

english

File:

PDF, 576 KB

english, 2008

6

The novel C-5 aryl, alkenyl, and alkynyl substituted uracil derivatives of l-ascorbic acid: Synthesis, cytostatic, and antiviral activity evaluations

Tatjana Gazivoda, Silvana Raić-Malić, Marko Marjanović, Marijeta Kralj, Krešimir Pavelić, Jan Balzarini, Erik De Clercq, Mladen Mintas

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 220 KB

english, 2007

7

Synthesis and antiviral activity of new pyrazole and thiazole derivatives

Osama I. El-Sabbagh, Mohamed M. Baraka, Samy M. Ibrahim, Christophe Pannecouque, Graciela Andrei, Robert Snoeck, Jan Balzarini, Adel A. Rashad

Journal:

European Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 268 KB

english, 2009

8

Synthesis, antimicrobial and antiviral evaluation of substituted imidazole derivatives

Deepika Sharma, Balasubramanian Narasimhan, Pradeep Kumar, Vikramjeet Judge, Rakesh Narang, Erik De Clercq, Jan Balzarini

Journal:

European Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 225 KB

english, 2009

9

Synthesis and Evaluation of Novel Acyclovir Phosphoramidates as Anti-HIV Agents

Davide Carta, Christopher McGuigan, Leonid Margolis, Jan Balzarini

Journal:

Antiviral Research

Year:

2009

Language:

english

File:

PDF, 88 KB

english, 2009

10

Design, synthesis and biological evaluation of cycloalkyl arylpyrimidines (CAPYs) as HIV-1 NNRTIs

Shuang-Xi Gu, Shi-Qiong Yang, Qiu-Qin He, Xiao-Dong Ma, Fen-Er Chen, Hui-Fang Dai, Erik De Clercq, Jan Balzarini, Christophe Pannecouque

Journal:

Bioorganic & Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 478 KB

english, 2011

11

Antiviral activity of carbohydrate-binding agents and the role of DC-SIGN in dengue virus infection

Marijke M.F. Alen, Suzanne J.F. Kaptein, Tine De Burghgraeve, Jan Balzarini, Johan Neyts, Dominique Schols

Journal:

Year:

2009

Language:

english

File:

PDF, 987 KB

english, 2009

12

Differential inhibition of various deoxyribonucleic acid polymerases by Evans blue and aurintricarboxylic acid

Hideo NAKANE, Jan BALZARINI, Erik de CLERCQ, Katsuhiko ONO

Journal:

Year:

1988

Language:

english

File:

PDF, 561 KB

english, 1988

13

The Application of Phosphoramidate Protide Technology to Acyclovir Confers Anti-HIV Inhibition

Derudas, Marco, Carta, Davide, Brancale, Andrea, Vanpouille, Christophe, Lisco, Andrea, Margolis, Leonid, Balzarini, Jan, McGuigan, Christopher

Journal:

Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 3.37 MB

english, 2009

14

Rational Design of 5‘-Thiourea-Substituted α-Thymidine Analogues as Thymidine Monophosphate Kinase Inhibitors Capable of Inhibiting Mycobacterial Growth

Van Daele, Ineke, Munier-Lehmann, Hélène, Froeyen, Matheus, Balzarini, Jan, Van Calenbergh, Serge

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 405 KB

english, 2007

15

5-chloro-substituted derivatives of 2',3'-didehydro-2' ,3'-dideoxyuridine, 3'-fluoro-2' ,3'-dideoxyuridine and 3'-azido-2' ,3'-dideoxyuridine as anti-HIV agents

Jan Balzarini, Arthur Van Aerschot, Piet Herdewijn, Erik De Clercq

Journal:

Biochemical Pharmacology

Year:

1989

Language:

english

File:

PDF, 574 KB

english, 1989

16

Activity and Safety of Synthetic Lectins Based on Benzoboroxole-Functionalized Polymers for Inhibition of HIV Entry

Mahalingam, Alamelu, Geonnotti, Anthony R., Balzarini, Jan, Kiser, Patrick F.

Journal:

Molecular Pharmaceutics

Year:

2011

Language:

english

File:

PDF, 3.63 MB

english, 2011

17

A Microwave-Assisted Diastereoselective Multicomponent Reaction To Access Dibenzo[ c , e ]azepinones: Synthesis and Biological Evaluation

Mehta, Vaibhav P., Modha, Sachin G., Ruijter, Eelco, Van Hecke, Kristof, Van Meervelt, Luc, Pannecouque, Christophe, Balzarini, Jan, Orru, Romano V. A., Van der Eycken, Erik

Journal:

Journal of Organic Chemistry

Year:

2011

Language:

english

File:

PDF, 2.22 MB

english, 2011

18

Synthesis and antiviral activity of monofluorinated cyclopropanoid nucleosides

Rosen, Thomas C., De Clercq, Erik, Balzarini, Jan, Haufe, G�nter

Journal:

Organic & Biomolecular Chemistry

Year:

2004

Language:

english

File:

PDF, 230 KB

english, 2004

19

Synthesis and Anti-herpetic Activity of Phosphoramidate ProTides

Maiti, Munmun, Persoons, Leentje, Andrei, Graciela, Snoeck, Robert, Balzarini, Jan, Herdewijn, Piet

Journal:

Year:

2013

Language:

english

File:

PDF, 526 KB

english, 2013

20

Phosphoramidate ProTides of the Anticancer Agent FUDR Successfully Deliver the Preformed Bioactive Monophosphate in Cells and Confer Advantage over the Parent Nucleoside

McGuigan, Christopher, Murziani, Paola, Slusarczyk, Magdalena, Gonczy, Blanka, Vande Voorde, Johan, Liekens, Sandra, Balzarini, Jan

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 2.05 MB

english, 2011

21

Synthesis and antiviral activity of highly water-soluble polycarboxylic derivatives of [70]fullerene

Kornev, Alexey B., Peregudov, Alexander S., Martynenko, Vyacheslav M., Balzarini, Jan, Hoorelbeke, Bart, Troshin, Pavel A.

Journal:

Chemical Communications

Year:

2011

Language:

english

File:

PDF, 1.08 MB

english, 2011

22

From norbornane-based nucleotide analogs locked in South conformation to novel inhibitors of feline herpes virus

Dejmek, Milan, Hřebabecký, Hubert, Šála, Michal, Dračínský, Martin, Procházková, Eliška, Leyssen, Pieter, Neyts, Johan, Balzarini, Jan, Nencka, Radim

Journal:

Bioorganic & Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 680 KB

english, 2014

23

Synthesis of triterpenoid triazine derivatives from allobetulone and betulonic acid with biological activities

Dinh Ngoc, Thuc, Moons, Nico, Kim, Youngju, De Borggraeve, Wim, Mashentseva, Anastassiya, Andrei, Graciela, Snoeck, Robert, Balzarini, Jan, Dehaen, Wim

Journal:

Bioorganic & Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 1000 KB

english, 2014

24

Application of ProTide Technology to Gemcitabine: A Successful Approach to Overcome the Key Cancer Resistance Mechanisms Leads to a New Agent (NUC-1031) in Clinical Development

Slusarczyk, Magdalena, Lopez, Monica Huerta, Balzarini, Jan, Mason, Malcolm, Jiang, Wen G., Blagden, Sarah, Thompson, Emely, Ghazaly, Essam, McGuigan, Christopher

Journal:

Journal of Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 1.32 MB

english, 2014

25

Synthesis of 5-Amino-3,3-dimethyl-7-phenyl-3 H -[1,2]oxathiolo[4,3- b ]pyridine-6-carbonitrile 1,1-Dioxides

Chioua, Mourad, Samadi, Abdelouahid, Postel, Denis, Balzarini, Jan, Marco-Contelles, José

Journal:

Journal of Heterocyclic Chemistry

Year:

2014

Language:

english

File:

PDF, 375 KB

english, 2014

26

Design and Discovery of a Novel Dipeptidyl-peptidase IV (CD26)-Based Prodrug Approach

García-Aparicio, Carlos, Bonache, María-Cruz, De Meester, Ingrid, San-Félix, Ana, Balzarini, Jan, Camarasa, María-José, Velázquez, Sonsoles

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 281 KB

english, 2006

27

Synthesis and Biological Evaluation of a Series of Substituted 2-Pyridine C-Nucleosides

Belmans, Marc, Esmans, Eddy, Dommisse, Roger, Lepoivre, Jozef, Alderweireldt, Frank, Balzarini, Jan, De Clercq, Erik

Journal:

Nucleosides and Nucleotides

Year:

1985

Language:

english

File:

PDF, 603 KB

english, 1985

28

Characterization of the activation pathway of phosphoramidate triester prodrugs of stavudine and zidovudine.

Saboulard, Didier, Naesens, Lieve, Cahard, Dominique, Salgado, Antonio, Pathirana, Ranjith, Velazquez, Sonsoles, McGuigan, Christopher, {De Clercq}, Erik, Balzarini, Jan

Journal:

Molecular Pharmacology

Year:

1999

Language:

english

File:

PDF, 212 KB

english, 1999

29

The ProTide Prodrug Technology: From the Concept to the Clinic

Mehellou, Youcef, Rattan, Hardeep S, Balzarini, Jan

Journal:

Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 3.89 MB

english, 2017

30

Nucleotide Delivery from cycloSaligenyl-3′-azido-3′-deoxythymidine Monophosphates (cycloSal-AZTMP)

Chris Meier, Eric De Clercq, Jan Balzarini

Journal:

European Journal of Organic Chemistry

Year:

1998

Language:

english

File:

PDF, 560 KB

english, 1998

31

Synthesis and Antiviral and Cytostatic Activities of Carbocyclic Nucleosides Incorporating a Modified Cyclobutane Ring

M. José Figueira, J. Manuel Blanco, Olga Caamaño, Franco Fernández, Xerardo García-Mera, Carmen López, Graciela Andrei, Robert Snoeck, Elisabeth Padalko, Johan Neyts, Jan Balzarini, Erik De Clercq

Journal:

Archiv der Pharmazie

Year:

1999

Language:

english

File:

PDF, 81 KB

english, 1999

32

Synthesis of 3-Nitrosoimidazo[1,2-a]pyridine Derivatives as Potential Antiretroviral Agents

Aziz Chaouni-Benabdallah, Christophe Galtier, Hassan Allouchi, Abdelhak Kherbeche, Jean-Claude Debouzy, Jean-Claude Teulade, Olivier Chavignon, Myriam Witvrouw, Christophe Pannecouque, Jan Balzarini,

Journal:

Archiv der Pharmazie

Year:

2001

Language:

english

File:

PDF, 91 KB

english, 2001

33

1,2,4-Triazole Derivatives Inhibiting the Human Immunodeficiency Virus Type 1 (HIV-1) in vitro

Irene M. Lagoja, Christophe Pannecouque, Laura Musumeci, Matheus Froeyen, Arthur Van Aerschot, Jan Balzarini, Piet Herdewijn, Erik De Clercq

Journal:

Helvetica Chimica Acta

Year:

2002

Language:

english

File:

PDF, 150 KB

english, 2002

34

Pridine Oxide Derivatives: Structure-Activity Relationship for Inhibition of Human Immunodeficiency Virus and Cytomegalovirus Replication in Cell Culture

Jan Balzarini, Miguel Stevens, Graciela Andrei, Robert Snoeck, Richard Strunk, James B. Pierce, John A. Lacadie, Erik De Clercq, Christophe Pannecouque

Journal:

Helvetica Chimica Acta

Year:

2002

Language:

english

File:

PDF, 135 KB

english, 2002

35

Palladium-Catalyzed Aryl Amination Reactions of 6-Bromo- and 6-Chloropurine Nucleosides

Paul F. Thomson, Pallavi Lagisetty, Jan Balzarini, Erik De Clercq, Mahesh K. Lakshman

Journal:

Advanced Synthesis & Catalysis

Year:

2010

Language:

english

File:

PDF, 225 KB

english, 2010

36

Bioreversible Maskierung von Nucleosiddiphosphaten

Henning Jacob Jessen, Tilmann Schulz, Jan Balzarini, Chris Meier

Journal:

Angewandte Chemie

Year:

2008

Language:

german

File:

PDF, 335 KB

german, 2008

37

Bioreversible Protection of Nucleoside Diphosphates

Henning Jacob Jessen, Tilmann Schulz, Jan Balzarini, Chris Meier

Journal:

Angewandte Chemie International Edition

Year:

2008

Language:

english

File:

PDF, 335 KB

english, 2008

38

Assessment of the in vitro broad-spectrum antiviral activity of some selected antitumor metallocene and metallocenium complexes

Sarah G Ward, R Craig Taylor, Petra Köpf-Maier, Hartmut Köpf, Jan Balzarini, Erik De Clercq

Journal:

Applied Organometallic Chemistry

Year:

1989

Language:

english

File:

PDF, 540 KB

english, 1989

39

Assessment of the in vitro broad-spectrum antiviral activity of some selected antitumor organotin complexes

Sarah G Ward, R Craig Taylor, Alan J Crowe, Jan Balzarini, Erik De Clercq

Journal:

Applied Organometallic Chemistry

Year:

1989

Language:

english

File:

PDF, 461 KB

english, 1989

40

Novel Carbocyclic Nucleosides Containing a Cyclopentyl Ring. Adenosine and Uridine Analogues

Carmen Balo, Franco Fernández, Evangelina Lens, Carmen López, Graciela Andrei, Robert Snoeck, Jan Balzarini, Erik De Clercq

Journal:

Archiv der Pharmazie

Year:

1997

Language:

english

File:

PDF, 339 KB

english, 1997

41

Non-nucleoside HIV Reverse Transcriptase Inhibitors, Part 6[1]: Synthesis and Anti-HIV Activity of Novel 2-[(Arylcarbonylmethyl)thio]-6-arylthio DABO Analogues

Guang-Fu Sun, Yun-Yan Kuang, Fen-Er Chen, Erik De Clercq, Jan Balzarini, Christophe Pannecouque

Journal:

Archiv der Pharmazie

Year:

2005

Language:

english

File:

PDF, 91 KB

english, 2005

42

Synthesis, Antiviral and Cytostatic Evaluation of Unsaturated Exomethylene and Keto D-Lyxopyranonucleoside Analogues

Niki Tzioumaki, Evangelia Tsoukala, Stella Manta, George Agelis, Jan Balzarini, Dimitri Komiotis

Journal:

Archiv der Pharmazie

Year:

2009

Language:

english

File:

PDF, 537 KB

english, 2009

43

Synthesis of 5′-N-(α-Amino-β-mercaptoacyl)amino-5′-deoxynucleosides as potential antiviral compounds

Rosario Herranz, Julia Castro-Pichel, M. Teresa García-López, Concepción Pérez, Jan Balzarini, Erik De Clercq

Journal:

Archiv der Pharmazie

Year:

1991

Language:

english

File:

PDF, 357 KB

english, 1991

44

Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors. Part 13 : Synthesis of Fluorine-Containing Diaryltriazine Derivatives for in vitro Anti-HIV Evaluation against Wild-Type Strain

Yuan-Zhen Xiong, Fen-Er Chen, Jan Balzarini, Erik De Clercq, Christophe Pannecouque

Journal:

Chemistry & Biodiversity

Year:

2009

Language:

english

File:

PDF, 194 KB

english, 2009

45

Non-Nucleoside HIV-1 Reverse-Transcriptase Inhibitors. Part 10 : Synthesis and Anti-HIV Activity of 5-Alkyl-6-(1-naphthylmethyl)pyrimidin-4(3H)-ones with a Mono- or Disubstituted 2-Amino Function as Novel ‘Dihydro-Alkoxy-Benzyl-Oxopyrimidine’ (DABO) Analogues

Yueping Wang, Fen-Er Chen, Jan Balzarini, Erik De Clercq, Christophe Pannecouque

Journal:

Chemistry & Biodiversity

Year:

2008

Language:

english

File:

PDF, 227 KB

english, 2008

46

Diastereoselective Synthesis of cycloSaligenyl-Nucleosyl-Phosphotriesters

Dr. Edwuin H. Rios Morales, Prof. Dr. Jan Balzarini, Prof. Dr. Chris Meier

Journal:

Chemistry - A European Journal

Year:

2011

Language:

english

File:

PDF, 406 KB

english, 2011

47

ChemInform Abstract: Lactate Cannot Substitute for Alanine in D4T-Based Anti-HIV Nucleotide Prodrugs — Despite Efficient Esterase-Mediated Hydrolysis.

Christopher McGuigan, Dominique Cahard, Carlo Ballatore, Adam Siddiqui, Erik De Clercq, Jan Balzarini

Journal:

Year:

1999

File:

PDF, 28 KB

1999

48

ChemInform Abstract: Synthesis and Biological Evaluation of Phosphonate Derivatives of Some Acyclic Pyridine-C-nucleosides.

Johan Van hemel, Eddy L. Esmans, Pieter E. Joos, Alex De Groot, Roger A. Dommisse, Jan M. Balzarini, Erik D. De Clercq

Journal:

Year:

1999

File:

PDF, 29 KB

1999

49

ChemInform Abstract: Synthesis and Biological Evaluation of a Carbocyclic Azanoraristeromycin Siderophore Conjugate.

Arun Ghosh, Marvin J. Miller, Erik De Clercq, Jan Balzarini

Journal:

Year:

1999

File:

PDF, 26 KB

1999

50

ChemInform Abstract: Synthesis and Antiviral Activity of Imidazo[1,2-a]pyridines.

Mohammed Lhassani, Olivier Chavignon, Jean-Michel Chezal, Jean-Claude Teulade, Jean-Pierre Chapat, Richard Snoeck, Graciela Andrei, Jan Balzarini, Erik De Clercq, Alain Gueiffier

Journal:

Year:

1999

File:

PDF, 28 KB

1999